SPR Methodologies to Advance Early Small-Molecule Programs for Challenging Membrane Protein Targets

  • Address key obstacles in SPR analysis of membrane proteins, including protein instability on the sensing surface and interference from detergent micelles
  • Showcase strategies for optimal detergent selection and membrane-protein stabilization to preserve activity during SPR experiments
  • Demonstrate how these optimized conditions enable reliable interaction profiling between small molecules and diverse membrane-protein classes